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Sarpogrelate hydrochloride
CAS No. 135159-51-2
Sarpogrelate hydrochloride ( MCI 9042;MCI9042;MCI-9042 )
产品货号. M11420 CAS No. 135159-51-2
A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥332 | 有现货 |
|
| 10MG | ￥535 | 有现货 |
|
| 25MG | ￥988 | 有现货 |
|
| 50MG | ￥1580 | 有现货 |
|
| 100MG | ￥2333 | 有现货 |
|
| 500MG | ￥5573 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Sarpogrelate hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
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产品描述A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.Heart Failure Approved
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同义词MCI 9042;MCI9042;MCI-9042
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通路Endocrinology/Hormones
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靶点5-HT Receptor
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受体5-HT Receptor
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研究领域Cardiovascular Disease
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适应症——
化学信息
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CAS Number135159-51-2
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分子量465.97
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分子式C24H32ClNO6
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纯度>98% (HPLC)
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溶解度DMSO: ≥ 62 mg/mL
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SMILESCN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl
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化学全称Butanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1)
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.
产品手册
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