Sarpogrelate hydrochloride ( MCI 9042;MCI9042;MCI-9042 )

产品货号. M11420 CAS No. 135159-51-2

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.

纯度: >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

规格	价格/人民币	库存	数量
5MG	￥332	有现货
10MG	￥535	有现货
25MG	￥988	有现货
50MG	￥1580	有现货
100MG	￥2333	有现货
500MG	￥5573	有现货
1G	获取报价	有现货

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生物学信息

产品名称

Sarpogrelate hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B.
产品描述

A potent, specific 5HT2 receptor antagonist with Ki of 8.39 nM for 5-HT2A; also shows binding affinity for 5-HT2B; displays selectivity over 5-HT1-like, 5-HT3, beta, H1, H2 and M3; blocks serotonin-induced platelet aggregation.Heart Failure Approved
同义词

MCI 9042;MCI9042;MCI-9042
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT Receptor
研究领域

Cardiovascular Disease
适应症

——

化学信息

CAS Number

135159-51-2
分子量

465.97
分子式

C24H32ClNO6
纯度

>98% (HPLC)
溶解度

DMSO: ≥ 62 mg/mL
SMILES

CN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl
化学全称

Butanedioic acid, 1-[2-(dimethylamino)-1-[[2-[2-(3-methoxyphenyl)ethyl]phenoxy]methyl]ethyl] ester, hydrochloride (1:1)

运输与储存

储存条件

(-20℃)
运输条件

With Ice Pack
稳定性

≥ 2 years

参考文献

1. Kikumoto R, et al. J Med Chem. 1990 Jun;33(6):1818-23.
2. Pertz H, et al. J Pharm Pharmacol. 1995 Apr;47(4):310-6.
3. Nishio H, et al. Arch Int Pharmacodyn Ther. 1996 Mar-Apr;331(2):189-202.

计算器

浓度计算器

摩尔计算器

分子量计算器

产品手册

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